Project ID CM-HD2026_21

ThemeCM-HD

Co Supervisor 1A Prof Maria R Sasi Conte Faculty of Dentistry, Oral & Craniofacial Sciences, Centre for Host-Microbiome InteractionsEmail

Co Supervisor 1B Prof Agamemnon E Grigoriadis Faculty of Dentistry, Oral & Craniofacial Sciences, Centre for Host-Microbiome InteractionsEmail

RNA binding protein regulation of cancer cell metabolism and tumorigenesis

Cancer cells have altered metabolism to cope with high energy demands associated with cell proliferation, migration and survival. The Conte and Grigoriadis labs explore the use of metabolic profiling, transcriptomics and proteomics to elucidate the role of two RNA binding proteins, LARP4A and LARP4B, that are key regulators of cancer cell behaviour and tumour progression.

We recently demonstrated that silencing of LARP4A and 4B inhibits cancer cell properties in vitro, and reduces tumour formation in xenograft models in vivo. LARP4A and 4B regulate the translation of a subset of mRNAs but the full list of target RNAs regulated by each LARP4 protein and the mechanisms linking mRNA translation regulation, cancer cell behaviour and tumourigenesis is not known. We have used NMR-based metabolomics, cell bioenergetics and RNAseq analyses of LARP4A/B-depleted cancer cells to identify the metabolic and signalling pathways affected by these proteins, and multiomics analysis identified targets involving hypoxia and glycolysis that are perturbed in knockdown cells. Moreover, LARP4A and LARP4B deletion appears to show differential cellular response at mitochondrial level. In this project the student will be trained in complementary skills of both Conte and Grigoriadis labs, including RNA structural biology, cancer cell biology and in vivo technology to achieve the following goals:

Year 1: Perform metabolomics, respirometry and proteomics profiles of cancer cell lines under different stress conditions (hypoxia, starvation) that are depleted in LARP4A and/or LARP4B using siRNA and CRISPR/Cas9 technologies. Experiments will be analysed by targeted and untargeted profiling for analysis of global changes.
Year 2: Validation of selected dysregulated genes, analyse metabolic profiles and function following small molecule inhibition and selected mutagenesis.
Years 2-3: Functional investigation of targets in vivo using multiple xenograft transplantation approaches; molecular analysis of LaRP4A/B RNA target interactions and write-up.
These studies will shed light for the first time on the mechanisms underlying the cancer-related functions of LARP4A and LARP4B.

During the rotation the student will focus on metabolism analysis of MG63 osteosarcoma cells, and how this is affected by sliencing LaRP4A/B proteins. Techiques will include cell biology, western blotting, respirometry and omics analysis. Details will be worked out with the student and will depend on latest data generated in the labs.

Representative Publications

1. Coleman JC, Hallett SR, Grigoriadis AE, Conte MR*. (2023) LARP4A and LARP4B in cancer: the new kids on the block – nt J Biochem Cell Biol. 161:106441. doi: 10.1016/j.biocel.2023.106441.
2. Cruz-Gallardo, I., Martino, L., Kelly, G., Atkinson, A., Trotta, R., De Tito, S., Coleman, P., Ahdash, Z., Gu, Y., Bui, T.TT Conte, M.R.* (2019) LARP4A recognises polyA RNA via a novel binding mechanism mediated by disordered regions and involving the PAM2w motif, revealing interplay between PABP, LARP4A and mRNA. Nucleic Acids Res., 47:4272-4291, doi: 10.1093/nar/gkz144
3. Graziani. V., Garcia, A.R,, Alcolado, L.S., Le Guennec, A., Henriksson, M.A.*, Conte, M.R.* (2023) Metabolic rewiring in MYC-driven medulloblastoma by BET-bromodomain inhibition. Sci Rep 13:1273. doi: 10.1038/s41598-023-27375-z

1. Coleman JC, Tattersall L, Yianni V, Knight L, Yu H, Hallett SR, Johnson P, Caetano A, Cosstick C, Ridley A, Gartland A, Conte MR*, Grigoriadis AE*. The RNA binding proteins LARP4A and LARP4B promote sarcoma and carcinoma growth and metastasis iScience. 2024, 27(4):109288. doi: 10.1016/j.isci.2024.109288
2. Weekes D, Kashima TG, Zandueta C, Perurena N, Thomas DP, Sunters A, Vuillier C, Bozec A, El-Emir E, Miletich I, Patiño-Garcia A, Lecanda F, Grigoriadis AE. (2016) Regulation of osteosarcoma cell lung metastasis by the c-Fos/AP-1 target FGFR1. Oncogene 35:2853
3. Cottone L, Ligammari L, Lee HM, Knowles HJ, Henderson S, Bianco S, Davies C, Strauss S, Amary F, Leite AP, Tirabosco R, Haendler K, Schultze JL, Herrero J, O’Donnell P, Grigoriadis AE, Salomoni P, Flanagan A. (2022). Aberrant paracrine signalling for bone remodelling underlies the mutant histone-driven giant cell tumour of bone. Cell Death Differ 29:2459. doi: 10.1038/s41418-022-01031-x